Umbralisib hydrochloride

Umbralisib hydrochloride

Cat Number
API1532533780
CAS Number
1532533-78-0

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CAS Number
1532533-78-0
Storage
Powder: -20℃ for 3 years. In solvent: -80℃ for 1 year.
Synonyms
RP5264 hydrochloride, TGR-1202 hydrochloride
Description
Umbralisib hydrochloride is a novel PI3Kδ inhibitor (IC50 and EC50 of 22.2 nM and 24.3 nM, respectively). Umbralisib hydrochloride is also active against CK1ε (EC50: 6.0 μM).
Molecular Formula
C31H25ClF3N5O3
Molecular Weight
608.01
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