Ponatinib D8 is a deuterium labeled Ponatinib. Ponatinib is an orally active inhibitor of multi-targeted kinase(Abl, PDGFRα, VEGFR2, FGFR1, and Src with IC50s of 0.37 nM, 1.1 nM, 1.5 nM, 2.2 nM, and 5.4 nM, respectively).
Molecular Formula
C29H27F3N6O
Molecular Weight
540.61
Storage
Powder: -20℃ for 3 years. In solvent: -80℃ for 1 year.