Taltirelin

Taltirelin

Cat Number
API103300749
CAS Number
103300-74-9

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CAS Number
103300-74-9
Synonyms
Taltirelin Acetate Ceredist TA 0910
Description
Taltirelin is a thyrotropin-releasing hormone receptor (TRH-R) superagonist with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Molecular Formula
C17H23N7O5
Molecular Weight
405.4
Appearance
White Solid
Melting Point
72-75℃
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