Rucaparib acetate

Rucaparib acetate

Cat Number
API773059237
CAS Number
773059-23-7

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CAS Number
773059-23-7
Description
Rucaparib (AG014699) acetate is a highly effective oral inhibitor of PARP proteins, specifically targeting PARP-1, PARP-2, and PARP-3, with a Ki value of 1.4 nM for PARP1. Additionally, it exhibits inhibitory action on hexose-6-phosphate dehydrogenase (H6PD) to a moderate extent. Rucaparib acetate shows promise in the field of research for castration-resistant prostate cancer (CRPC).
Molecular Formula
C21H22FN3O3
Molecular Weight
383.423
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