Alpelisib hydrochloride

Alpelisib hydrochloride

Cat Number
API1584128915
CAS Number
1584128-91-5

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CAS Number
1584128-91-5
Storage
Powder: -20℃ for 3 years. In solvent: -80℃ for 1 year.
Description
Alpelisib hydrochloride (BYL-719 hydrochloride) exhibits anticancer properties. As a potent and selective PI3Kα inhibitor with high oral bioavailability, it has IC50 values of 5 nM for p110α, 250 nM for p110γ, 290 nM for p110δ, and 1200 nM for p110β, indicating its efficacy in targeting enzymes involved in cancer cell proliferation.
Molecular Formula
C19H23ClF3N5O2S
Molecular Weight
477.93
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