Umbralisib hydrochloride is a novel PI3Kδ inhibitor (IC50 and EC50 of 22.2 nM and 24.3 nM, respectively). Umbralisib hydrochloride is also active against CK1ε (EC50: 6.0 μM).
Molecular Formula
C31H25ClF3N5O3
Molecular Weight
608.01
Storage
Powder: -20℃ for 3 years. In solvent: -80℃ for 1 year.