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Cat Number: API2062784

PimozideR6238

CAS Number

2062-78-4

Description

Pimozide (R6238) is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic receptors in the central nervous system (CNS), thereby decreasing dopamine neurotransmission and reducing the occurrence of the motor and vocal tics and delusions of parasitosis. In addition, this agent antagonizes alpha-adrenergic and 5-HT2 receptors.

Molecular Formula

C28H29F2N3O

Molecular Weight

461.55

Smiles

FC1CCC(CC1)C(CCCN1CCC(CC1)N1C2CCCCC2[NH]C1=O)C1CCC(F)CC1

Purity

Storage

Powder: -20℃ for 3 years. In solvent: -80℃ for 1 year.

Solubility Information

DMSO: 6 mg/mL (13 mM)

Relative Density