Lapatinib tosylate

Lapatinib tosylate

Cat Number
API1187538357
CAS Number
1187538-35-7

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CAS Number
1187538-35-7
Synonyms
GW2016 tosylate
Description
Lapatinib tosylate (GW572016), a robust and orally administered inhibitor specifically targeting the tyrosine kinase domains of ErbB-2 and EGFR, exhibits inhibitory concentration 50 (IC50) values of 10.2 nM and 9.8 nM against purified EGFR and ErbB-2, respectively.
Molecular Formula
C36H34ClFN4O7S2
Molecular Weight
753.26
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